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Directory

Small Molecule Drug Companies in the UK

Small molecule drug companies develop low-molecular-weight medicines designed to interact with specific biological targets. These compounds can often enter cells and may be formulated as oral or other conventional dosage forms across a wide range of therapeutic areas.

This category includes companies working on:

  • Small molecule drug discovery and screening
  • Medicinal chemistry and lead optimisation
  • Targeted inhibitors and molecular modulators
  • Preclinical development and candidate selection
  • Oral medicines and specialist drug formulations

Browse 202 UK small molecule drug companies below.

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Small Molecule Drugs
Showing 133–144 of 202
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Isomorphic Labs

Greater London

AI-powered drug design engine built on AlphaFold technology

Isomorphic Labs is an artificial intelligence company applying frontier AI to drug discovery, built on and beyond the Nobel Prize-winning AlphaFold protein structure prediction…

SoftwareBiotech
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Agility Life Sciences

Midlands

Formulation development CDMO for difficult pharmaceuticals

Agility Life Sciences is a contract development and manufacturing organisation specialising in pharmaceutical formulation development. Based in Stapleford, Nottingham, the company…

CDMO
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Vernalis

East of England

Fragment and structure-based drug discovery services

Vernalis (R&D) is a Cambridge-based contract drug discovery organisation specialising in fragment-based and structure-based drug discovery. The company integrates structural…

CROBiotech
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AstronauTx

Greater London

Small molecule drugs targeting astrocytes in neurodegenerative disease

AstronauTx is a clinical-stage UK biotech developing oral small molecule therapeutics for Alzheimer's disease and other neurodegenerative disorders. The company's approach targets…

Biotech
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Hikma Pharmaceuticals

Greater London

Global generics and specialty pharmaceutical manufacturer headquartered in London

Hikma Pharmaceuticals is a multinational pharmaceutical company developing, manufacturing and marketing generic, specialty and branded medicines across injectable, oral and…

Biopharma
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Tailor Bio

East of England

AI platform targeting chromosomal instability across cancer

Tailor Bio is a Cambridge-based biotechnology company developing an AI-driven precision medicine platform for cancers with chromosomal instability, a genomic phenomenon present in…

Biotech
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Enterprise Therapeutics

South East England

Small molecule therapies for cystic fibrosis and COPD

Enterprise Therapeutics is a clinical-stage biopharmaceutical company developing novel muco-regulatory therapies for respiratory diseases. Its lead programme ETD001 is a…

Biopharma
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Outrun Therapeutics

Scotland

E3 ligase inhibitors stabilising tumour suppressor proteins

Outrun Therapeutics is a preclinical drug discovery company developing small molecule inhibitors of E3 ligase enzymes to stabilise tumour suppressor and other disease-relevant…

Biotech
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Hypha Discovery

South East England

Specialist CRO for drug and agrochemical metabolite synthesis and characterisation

Hypha Discovery is a specialist contract research organisation supporting pharmaceutical and agrochemical companies worldwide. The company produces and purifies drug and…

CROReagents & Consumables
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Mission Therapeutics

East of England

DUB inhibitor therapeutics targeting mitophagy and degenerative disease

Mission Therapeutics is a clinical-stage biotechnology company developing first-in-class small molecule inhibitors of deubiquitylating enzymes to treat diseases driven by…

Biotech
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Pathios Therapeutics

South East England

Small molecule GPR65 inhibitors restoring immune response in solid tumours

Pathios Therapeutics is a clinical-stage drug discovery company developing small molecule inhibitors of GPR65, a pH-sensing G protein-coupled receptor that drives…

Biotech
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IngenOx Therapeutics

South East England

Precision oncology drugs and vaccines for cold tumours

IngenOx Therapeutics Limited is a clinical-stage biopharmaceutical company developing precision oncology drugs and cancer vaccines for difficult-to-treat tumours. The company…

BiotechBiopharma
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